Concepedia

Synthesis and biological evaluation of novel heterocyclic derivatives of combretastatin A-4

Thị Thanh Bình Nguyễn, Thierry Lomberget, Ngoc Chau Tran, Evelyne Colomb, Lore Nachtergaele, Sylviane Thoret, Joëlle Dubois, Joren Guillaume, Rawad Abdayem, Marek Haftek,

Bioorganic & Medicinal Chemistry Letters · 2012 · 33 citations · 34 references

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References

34

Normal keratinization in a spontaneously immortalized aneuploid human keratinocyte cell line.

Petra Boukamp, R T Petrussevska, Dirk Breitkreutz et al. · The Journal of Cell Biology · 1988 · 4.2K citations · Full text

, , +11

Isolation and structure of the strong cell growth and tubulin inhibitor combretastatin A-4

George R. Pettit, Sheo B. Singh, Ernest Hamel et al. · Cellular and Molecular Life Sciences · 1989 · 789 citations

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Potent, Orally Active Heterocycle-Based Combretastatin A-4 Analogues:  Synthesis, Structure−Activity Relationship, Pharmacokinetics, and In Vivo Antitumor Activity Evaluation

Le Wang, Keith W. Woods, Qun Li et al. · Journal of Medicinal Chemistry · 2002 · 421 citations · Full text

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Antineoplastic Agents. 291. Isolation and Synthesis of Combretastatins A-4, A-5, and A-6

George R. Pettit, Sheo B. Singh, Michael R. Boyd et al. · Journal of Medicinal Chemistry · 1995 · 391 citations

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Interactions of tubulin with potent natural and synthetic analogs of the antimitotic agent combretastatin: a structure-activity study.

C. Michael Lin, Sheo B. Singh, Ping S. Chu et al. · Molecular Pharmacology · 1988 · 282 citations

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