Ultra-High Throughput Screen of Two-Million-Member Combinatorial Compound Collection in a Miniaturized, 1536-Well Assay Format

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

Ji-Hu Zhang, Thomas D.Y. Chung, Kevin R. Oldenburg · SLAS DISCOVERY · 1999 · 7K citations · Full text

Pharmacy, Medicinal Chemistry, Drug Design +16

Strategy and Tactics in Combinatorial Organic Synthesis. Applications to Drug Discovery

Eric M. Gordon, Mark A. Gallop, Dinesh V. Patel · Accounts of Chemical Research · 1996 · 267 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +6

Assay Miniaturization for Ultra-High Throughput Screening of Combinatorial and Discrete Compound Libraries: A 9600-Well (0.2 Microliter) Assay System

Kevin R. Oldenburg, Ji-Hu Zhang, Tongming Chen et al. · SLAS DISCOVERY · 1998 · 73 citations · Full text

Pharmacy, Medicinal Chemistry, Combinatorial Chemistry +13

Identification of potent inhibitors of Plasmodium falciparum plasmepsin II from an encoded statine combinatorial library

Carolyn DiIanni Carroll, Hitesh D. Patel, Theodore Johnson et al. · Bioorganic & Medicinal Chemistry Letters · 1998 · 68 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

A High-Density Screening Format for Encoded Combinatorial Libraries: Assay Miniaturization and Its Application to Enzymatic Reactions

John R. Schullek, John H. Butler, Zhi‐Jie Ni et al. · Analytical Biochemistry · 1997 · 61 citations

Life Sciences, Biochemistry, Biotechnology +17