Concepedia

Pharmacophore elements of the TIPP class of delta opioid receptor antagonists

Henry I. Mosberg, John R. Omnaas, Katarzyna Sobczyk‐Kojiro, Raj Dua, Jeffrey C. Ho, Wenli Ma, Paula Bush, Carol Mousigian, Andrei L. Lomize

Letters in Peptide Science · 1994 · 20 citations · 7 references

DOI

Concepts

References

7

Application of the message-address concept in the design of highly potent and selective non-peptide .delta. opioid receptor antagonists

P. S. Portoghese, Marjia Sultana, Hiroshi Nagase et al. · Journal of Medicinal Chemistry · 1988 · 305 citations

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Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists.

Peter W. Schiller, Tin Nguyen, Grazyna Weltrowska et al. · Proceedings of the National Academy of Sciences · 1992 · 240 citations · Full text

, , +17

TIPP[.psi.]: a highly potent and stable pseudopeptide .delta. opioid receptor antagonist with extraordinary .delta. selectivity

Peter W. Schiller, Grazyna Weltrowska, Thi M.‐D. Nguyen et al. · Journal of Medicinal Chemistry · 1993 · 147 citations · Full text

, , +16

Selective Opioid Dipeptides

Piero Andrea Temussi, Severo Salvadori, Pietro Amodeo et al. · Biochemical and Biophysical Research Communications · 1994 · 86 citations

Cyclic, disulfide- and dithioether-containing opioid tetrapeptides: Development of a ligard with high delta opioid receptor selectivity and affinity

Henry I. Mosberg, John R. Omnaas, Fedor Medzihradsky et al. · Life Sciences · 1988 · 68 citations · Full text

, , +16