Grazyna Weltrowska

Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists.

Peter W. Schiller, Tin Nguyen, Grazyna Weltrowska et al. · Proceedings of the National Academy of Sciences · 1992 · 239 citations · Full text

Unprecedented Delta Selectivity, Pharmacotherapy, Opioid Peptide Analogs +18

The Opioid μ Agonist/δ Antagonist DIPP-NH₂[Ψ] Produces a Potent Analgesic Effect, No Physical Dependence, and Less Tolerance than Morphine in Rats

Peter W. Schiller, Marian E. Fundytus, Lisa Merovitz et al. · Journal of Medicinal Chemistry · 1999 · 186 citations · Full text

Opioid Epidemic, Pain Disorders, Pain Medicine +26

Synthesis and in vitro opioid activity profiles of DALDA analogues

Peter W. Schiller, Thi M.‐D. Nguyen, Irena Berezowska et al. · European Journal of Medicinal Chemistry · 2000 · 161 citations · Full text

Dalda Analogues, Pharmacological Study, Biochemistry +8

Attenuation of morphine tolerance and dependence with the highly selective δ-opioid receptor antagonist TIPP[ψ]

Marian E. Fundytus, Peter W. Schiller, M.M. Shapiro et al. · European Journal of Pharmacology · 1995 · 156 citations

Opioid Epidemic, Molecular Pharmacology, Morphine Tolerance +12

TIPP[.psi.]: a highly potent and stable pseudopeptide .delta. opioid receptor antagonist with extraordinary .delta. selectivity

Peter W. Schiller, Grazyna Weltrowska, Thi M.‐D. Nguyen et al. · Journal of Medicinal Chemistry · 1993 · 147 citations · Full text