Concepedia

The first synthetic agonists of FFA2: Discovery and SAR of phenylacetamides as allosteric modulators

Yingcai Wang, Xian‐Yun Jiao, Frank Kayser, Jiwen Liu, Zhongyu Wang, Malgorzata Wanska, Joanne Greenberg, Jennifer Weiszmann, Hongfei Ge, Hui Tian,

Bioorganic & Medicinal Chemistry Letters · 2009 · 100 citations · 12 references

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12

The Orphan G Protein-coupled Receptors GPR41 and GPR43 Are Activated by Propionate and Other Short Chain Carboxylic Acids

Andrew J. Brown, Susan M. Goldsworthy, Ashley Barnes et al. · Journal of Biological Chemistry · 2003 · 2.3K citations · Full text

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Functional Characterization of Human Receptors for Short Chain Fatty Acids and Their Role in Polymorphonuclear Cell Activation

Emmanuel Le Poul, Cécile Loison, Sofie Struyf et al. · Journal of Biological Chemistry · 2003 · 1.6K citations · Full text

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Acetate and Propionate Short Chain Fatty Acids Stimulate Adipogenesis via GPCR43

Yeon-Hee Hong, Yukihiko Nishimura, Daisuke Hishikawa et al. · Endocrinology · 2005 · 602 citations · Full text

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Identification of a free fatty acid receptor, FFA2R, expressed on leukocytes and activated by short-chain fatty acids

Niclas Nilsson, Knut Kotarsky, Christer Owman et al. · Biochemical and Biophysical Research Communications · 2003 · 540 citations

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Activation of G Protein-Coupled Receptor 43 in Adipocytes Leads to Inhibition of Lipolysis and Suppression of Plasma Free Fatty Acids

Hongfei Ge, Xiaofan Li, Jennifer Weiszmann et al. · Endocrinology · 2008 · 470 citations · Full text

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