Concepedia

Peptide-derived transition state analogue inhibitors of thrombin; Synthesis, activity and selectivity

Mieke Jetten, Co A.M. Peters, Arie Visser, Peter D. J. Grootenhuis, J. W. VAN NISPEN, H. C. J. OTTENHEIJM

Bioorganic & Medicinal Chemistry · 1995 · 13 citations · 39 references

DOI

Concepts

References

39

On the size of the active site in proteases. I. Papain

Israël Schechter, Arieh Berger · Biochemical and Biophysical Research Communications · 1967 · 5.2K citations

, , +9

Comprehensive medicinal chemistry

H. Timmerman, Aalt Bast, H. van der Goot et al. · Trends in Pharmacological Sciences · 1991 · 1.2K citations

The refined 1.9 A crystal structure of human alpha‐thrombin: interaction with D‐Phe‐Pro‐Arg chloromethylketone and significance of the Tyr‐Pro‐Pro‐Trp insertion segment.

Wolfram Bode, Irmgard Mayr, Ulrich Baumann et al. · The EMBO Journal · 1989 · 893 citations · Full text

, , +6

Molecular Architecture and
\nBiological Reactions

Linus Pauling · CaltechAUTHORS (California Institute of Technology) · 1946 · 854 citations

, , +8

Peptides: Chemistry, structure and biology

Rebecca C. Wade · FEBS Letters · 1977 · 840 citations

, , +10