Concepedia

Design and synthesis of guanylthiourea derivatives as potential inhibitors of Plasmodium falciparum dihydrofolate reductase enzyme

Legesse Adane, Shweta Bhagat, Minhajul Arfeen, Sonam Bhatia, Rachada Sirawaraporn, Worachart Sirawaraporn, Asit K. Chakraborti, Prasad V. Bharatam

Bioorganic & Medicinal Chemistry Letters · 2013 · 39 citations · 33 references

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33

Glide:  A New Approach for Rapid, Accurate Docking and Scoring. 1. Method and Assessment of Docking Accuracy

Richard A. Friesner, Jay L. Banks, Robert B. Murphy et al. · Journal of Medicinal Chemistry · 2004 · 9.9K citations

, , +17

Glide:  A New Approach for Rapid, Accurate Docking and Scoring. 2. Enrichment Factors in Database Screening

Thomas A. Halgren, Robert B. Murphy, Richard A. Friesner et al. · Journal of Medicinal Chemistry · 2004 · 5.2K citations

, , +17

Minimization of variation in the response to different proteins of the Coomassie blue G dye-binding assay for protein

Steve M. Read, D. H. Northcote · Analytical Biochemistry · 1981 · 1.4K citations

, , +11

Amino acid changes linked to pyrimethamine resistance in the dihydrofolate reductase-thymidylate synthase gene of Plasmodium falciparum.

Alan F. Cowman, M J Morry, Beverley‐Ann Biggs et al. · Proceedings of the National Academy of Sciences · 1988 · 530 citations · Full text

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Insights into antifolate resistance from malarial DHFR-TS structures

Jirundon Yuvaniyama, P. Chitnumsub, Sumalee Kamchonwongpaisan et al. · Nature Structural & Molecular Biology · 2003 · 411 citations · Full text

, , +14