Bioorganic & Medicinal Chemistry Letters · 2012 · 118 citations · 1 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryEnzymologyEnzyme DiscoveryEnzyme InhibitionHit-to-lead OptimizationPotency OptimizationTopoisomerase InhibitorsCatalytic Topoisomerase InhibitionPyrimidine AnalogsPyrimidine AnaloguesPyrimidine ChemistryStructure-based Enzyme TargetingTopoisomerase Activity
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