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The design and synthesis of thrombin inhibitors: analogues of MD805 containing non-polar surrogates for arginine at the P1 position

Urs Baettig, Lyndon Brown, Derek E. Brundish, C. P. Dell, Alex Furzer, Sheila Garman, Diana Janus, Peter D. Kane, Garrick Smith, Clive V Walker,

Bioorganic & Medicinal Chemistry Letters · 2000 · 13 citations · 6 references

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6

Thionation reactions of lawesson's reagents

Michael P. Cava, Matthew I. Levinson · Tetrahedron · 1985 · 661 citations

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Thrombin inhibitors. 3. Carboxyl-containing amide derivatives of N.alpha.-substituted L-arginine

Ryoji Kikumoto, Y Tamao, Kazuo Ohkubo et al. · Journal of Medicinal Chemistry · 1980 · 51 citations · Full text

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Thrombin inhibitors. 1. Ester derivatives of N.alpha.-(arylsulfonyl)-L-arginine

Shosuke Okamoto, Kiyokatsu Kinjo, Akiko Hijikata et al. · Journal of Medicinal Chemistry · 1980 · 49 citations · Full text

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Synthesis of a novel class of heteroaromatic amino acids and their use in the preparation of analogs of luteinizing hormone-releasing hormone

John J. Nestor, Bonnie L. Horner, Teresa L. Ho et al. · Journal of Medicinal Chemistry · 1984 · 34 citations

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Argatroban analogs: Synthesis, thrombin inhibitory activity and cell permeability of aminoheterocyclic guanidine surrogates

Raj N. Misra, Yolanda F. Kelly, Bärbel R. Brown et al. · Bioorganic & Medicinal Chemistry Letters · 1994 · 32 citations

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