Concepedia

Publication | Open Access

Participation of CYP2C8 and CYP3A4 in the N‐demethylation of imatinib in human hepatic microsomes

87

Citations

36

References

2010

Year

Abstract

CYP2C8 and CYPs 3A contribute to imatinib N-demethylation in human liver. The involvement of CYP2C8 may account in part for the wide inter-patient variation in imatinib pharmacokinetics observed in clinical practice.

References

YearCitations

Page 1