Teresa W. Makowski

Use of an Iridium-Catalyzed Redox-Neutral Alcohol-Amine Coupling on Kilogram Scale for the Synthesis of a GlyT1 Inhibitor

Martin A. Berliner, Stéphane Dubant, Teresa W. Makowski et al. · Organic Process Research & Development · 2011 · 110 citations

Natural Sciences, Chemistry, Medicinal Chemistry +10

Commercial Route Research and Development for SGLT2 Inhibitor Candidate Ertugliflozin

Paul Bowles, Steven J. Brenek, Stéphane Caron et al. · Organic Process Research & Development · 2013 · 67 citations

Pharmacy, Medicinal Chemistry, Pharmacology +9

Developing an Asymmetric Transfer Hydrogenation Process for (<i>S</i>)-5-Fluoro-3-methylisobenzofuran-1(3<i>H</i>)-one, a Key Intermediate to Lorlatinib

Shengquan Duan, Bryan Li, Robert W. Dugger et al. · Organic Process Research & Development · 2017 · 35 citations

Natural Sciences, Chemistry, Medicinal Chemistry +14

Synthesis of 1,2,3,4-Tetrahydroisoquinolines Containing Electron-Withdrawing Groups

George J. Quallich, Teresa W. Makowski, Andrew F. Sanders et al. · The Journal of Organic Chemistry · 1998 · 35 citations

Natural Sciences, Chemistry, Medicinal Chemistry +7

Investigation of Practical Routes for the Kilogram-Scale Production of <i>cis</i>-3-Methylamino-4-methylpiperidines

Weiling Cai, James L. Colony, Heather N. Frost et al. · Organic Process Research & Development · 2005 · 29 citations

Natural Sciences, Chemistry, Medicinal Chemistry +14