Paul A. J. Janssen

Receptor binding profile of R 41 468, A novel antagonist at 5-HT2 receptors

J.E. Leysen, F. Awouters, Ludo Kennis et al. · Life Sciences · 1981 · 846 citations

Medicine, Medicinal Chemistry, Pharmacology +13

Potent and selective inhibition of HIV-1 replication in vitro by a novel series of TIBO derivatives

Rudi Pauwels, Koen Andries, Jan Desmyter et al. · Nature · 1990 · 757 citations

Medicine, Medicinal Chemistry, Pharmacology +12

Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 Variants

Kalyan Das, Arthur D. Clark, Paul Lewi et al. · Journal of Medicinal Chemistry · 2004 · 511 citations

Life Sciences, Medicinal Chemistry, Pharmacology +17

Pharmacology of risperidone (R 64 766), a new antipsychotic with serotonin-S2 and dopamine-D2 antagonistic properties.

Paul A. J. Janssen, C. J. E. Niemegeers, F. Awouters et al. · Journal of Pharmacology and Experimental Therapeutics · 1988 · 468 citations

Medicine, Pharmacology, Pharmacotherapy +14

Biochemical profile of risperidone, a new antipsychotic.

J.E. Leysen, W Gommeren, A Eens et al. · Journal of Pharmacology and Experimental Therapeutics · 1988 · 413 citations

Medicine, Pharmacology, Pharmacotherapy +17