Haiching Ma

Comprehensive assay of kinase catalytic activity reveals features of kinase inhibitor selectivity

Theonie Anastassiadis, Sean Deacon, Karthik Devarajan et al. · Nature Biotechnology · 2011 · 926 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +16

Human 3α-hydroxysteroid dehydrogenase isoforms (AKR1C1‒AKR1C4) of the aldo-keto reductase superfamily: functional plasticity and tissue distribution reveals roles in the inactivation and formation of male and female sex hormones

T.M. Penning, Michael E. Burczynski, Joseph M. Jez et al. · Biochemical Journal · 2000 · 572 citations · Full text

Life Sciences, Biochemistry, Endocrinology +17

Human 3α-hydroxysteroid dehydrogenase isoforms (AKR1C1–AKR1C4) of the aldo-keto reductase superfamily: functional plasticity and tissue distribution reveals roles in the inactivation and formation of male and female sex hormones

T.M. Penning, Michael E. Burczynski, Joseph M. Jez et al. · Biochemical Journal · 2000 · 350 citations

Life Sciences, Biochemistry, Endocrinology +17

Conformational Analysis of the DFG-Out Kinase Motif and Biochemical Profiling of Structurally Validated Type II Inhibitors

Ramachandran Vijayan, Peng He, Vivek Modi et al. · Journal of Medicinal Chemistry · 2014 · 245 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +14

The challenge of selecting protein kinase assays for lead discovery optimization

Haiching Ma, Sean Deacon, Kurumi Y. Horiuchi · Expert Opinion on Drug Discovery · 2008 · 200 citations · Full text

Pharmacy, Pharmaceutical Biotechnology, Drug Design +8