Scott Savage

Efficient Synthesis of 4-, 5-, and 6-Methyl-2,2‘-bipyridine by a Negishi Cross-Coupling Strategy Followed by High-Yield Conversion to Bromo- and Chloromethyl-2,2‘-bipyridines

Scott Savage, Adam P. Smith, Cassandra L. Fraser · The Journal of Organic Chemistry · 1998 · 111 citations

Cross-coupling Reaction, Engineering, Virginia 22901 +13

Highly Stereoselective Synthesis of Tetrasubstituted Acyclic All-Carbon Olefins via Enol Tosylation and Suzuki–Miyaura Coupling

Beryl X. Li, Diane N. Le, Andrew McClory et al. · Journal of the American Chemical Society · 2017 · 97 citations · Full text

Preparation of Saxagliptin, a Novel DPP-IV Inhibitor

Scott Savage, Gregory Jones, Sergei Kolotuchin et al. · Organic Process Research & Development · 2009 · 75 citations

Pharmaceutical Science, Bioorganic Chemistry, Organic Chemistry +16

Identification of <i>C</i>-2 Hydroxyethyl Imidazopyrrolopyridines as Potent JAK1 Inhibitors with Favorable Physicochemical Properties and High Selectivity over JAK2

Mark Zak, Christopher A. Hurley, Stuart I. Ward et al. · Journal of Medicinal Chemistry · 2013 · 61 citations · Full text

Pharmaceutical Science, Pharmacotherapy, Chemical Biology +19

Discovery and Optimization of <i>C</i>-2 Methyl Imidazopyrrolopyridines as Potent and Orally Bioavailable JAK1 Inhibitors with Selectivity over JAK2

Mark Zak, Rohan Mendonca, Mercedesz Balázs et al. · Journal of Medicinal Chemistry · 2012 · 61 citations · Full text

Pharmaceutical Science, Pharmacotherapy, Chemical Biology +16