Concepedia

Brad Newhouse

BN

Statistics

Publications

7

Citations

955

H-Index

7

Active since

2008

Affiliations

Array BioPharma (United States)(Current)

Brad Newhouse is an author at Array BioPharma (United States) specializing in medicinal chemistry, pharmacology, and drug discovery.

Publications per year

2008–2021

7

Publications

7

Identification of MRTX1133, a Noncovalent, Potent, and Selective KRAS <sup>G12D</sup> Inhibitor

Xiaolun Wang, Shelley Allen, James F. Blake et al. · Journal of Medicinal Chemistry · 2021 · 708 citations · Full text

, , +14

Pyrazolopyridine Inhibitors of B-Raf<sup>V600E</sup>. Part 1: The Development of Selective, Orally Bioavailable, and Efficacious Inhibitors

Steve Wenglowsky, Li Ren, Kateri A. Ahrendt et al. · ACS Medicinal Chemistry Letters · 2011 · 66 citations · Full text

, , +15

Potent and selective pyrazole-based inhibitors of B-Raf kinase

Joshua D. Hansen, Jonas Grina, Brad Newhouse et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 65 citations · Full text

, , +11

Pyrazolopyridine inhibitors of B-RafV600E. Part 2: Structure–activity relationships

Steve Wenglowsky, Kateri A. Ahrendt, Alex J. Buckmelter et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 56 citations · Full text

, , +13

Potent and selective pyrazolo[1,5-a]pyrimidine based inhibitors of B-RafV600E kinase with favorable physicochemical and pharmacokinetic properties

Li Ren, Ellen R. Laird, Alex J. Buckmelter et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 24 citations · Full text

, , +13

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