Lee D. Fader

Revealing Atropisomer Axial Chirality in Drug Discovery

Steven R. LaPlante, Paul Edwards, Lee D. Fader et al. · ChemMedChem · 2011 · 499 citations

Molecular Pharmacology, Medicinal Chemistry, Molecular Sciences +15

Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1

Lee D. Fader, Éric Malenfant, Mathieu Parisien et al. · ACS Medicinal Chemistry Letters · 2014 · 175 citations · Full text

Hiv-1 Integrase, Immunology, Molecular Biology +16

Distinct Effects of Two HIV-1 Capsid Assembly Inhibitor Families That Bind the Same Site within the N-Terminal Domain of the Viral CA Protein

Christopher T. Lemke, Steve Titolo, Uta von Schwedler et al. · Journal of Virology · 2012 · 124 citations · Full text

Arylcyclopropanes: Properties, Synthesis and Use in Medicinal Chemistry

Alexandre Gagnon, Martin Duplessis, Lee D. Fader · Organic Preparations and Procedures International · 2010 · 121 citations

Medicinal Chemistry, Unique Steric, Engineering +10

Discovery of a 1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione series of inhibitors of HIV-1 capsid assembly

Lee D. Fader, Richard C. Bethell, Pierre Bonneau et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 104 citations

Combinatorial Chemistry, Medicinal Chemistry, Heterocyclic +8