Intracellular repair of oxidation-damaged α-synuclein fails to target C-terminal modification sites

Andrés Binolfi, Antonio Limatola, Silvia Verzini, +7

Nature Communications

Synthesis, in Vitro, and in Cell Studies of a New Series of [Indoline-3,2′-thiazolidine]-Based p53 Modulators

Alessia Bertamino, Maria Soprano, Simona Musella, +12

Journal of Medicinal Chemistry

Chemoprevention StrategyP53 ProteinNew SeriesPharmaceutical ChemistryTumor Biology +15

Apoptosis Therapy in Cancer: The First Single-molecule Co-activating p53 and the Translocator Protein in Glioblastoma

Simona Daniele, Sabrina Taliani, Eleonora Da Pozzo, +13

Scientific Reports

Novel α-MSH Peptide Analogues with Broad Spectrum Antimicrobial Activity

Paolo Grieco, Alfonso Carotenuto, Luigia Auriemma, +11

PLoS ONE

Novel Cyclic Biphalin Analogue with Improved Antinociceptive Properties

Adriano Mollica, Alfonso Carotenuto, Ettore Novellino, +12

ACS Medicinal Chemistry Letters

Pain MedicineMolecular PainProducts 9PharmacotherapyPharmaceutical Chemistry +17

Time‐Resolved NMR Analysis of Proteolytic α‐Synuclein Processing in vitro and in cellulo

Antonio Limatola, Cédric Eichmann, Reeba S. Jacob, +4

PROTEOMICS

Lead Optimization of P5U and Urantide: Discovery of Novel Potent Ligands at the Urotensin-II Receptor

Alfonso Carotenuto, Luigia Auriemma, Francesco Merlino, +10

Journal of Medicinal Chemistry

Lead IdentificationImportant LigandsPharmacotherapyMedicinal ChemistryNovel Ligands +14

An investigation into the origin of the biased agonism associated with the urotensin II receptor activation

Diego Brancaccio, Francesco Merlino, Antonio Limatola, +6

Journal of Peptide Science

Biased AgonismUrotensin Ii ReceptorChemical BiologyCell SignalingMolecular Physiology +17

Design, synthesis and efficacy of novel G protein-coupled receptor kinase 2 inhibitors

Alfonso Carotenuto, Ersilia Cipolletta, Isabel Gómez‐Monterrey, +11

European Journal of Medicinal Chemistry

BiochemistryFunctional SelectivityMedicineG Protein-coupled ReceptorReceptor Tyrosine Kinase +5

Development of Macrocyclic Peptidomimetics Containing Constrained α,α-Dialkylated Amino Acids with Potent and Selective Activity at Human Melanocortin Receptors

Francesco Merlino, Yang Zhou, Minying Cai, +9

Journal of Medicinal Chemistry

Combinatorial ChemistryAmino AcidsMolecular BiologyMolecular PharmacologyMedicinal Chemistry +15