Synthesis, in Vitro, and in Cell Studies of a New Series of [Indoline-3,2′-thiazolidine]-Based p53 Modulators

Alessia Bertamino, Maria Soprano, Simona Musella, +12

Journal of Medicinal Chemistry

Chemoprevention StrategyP53 ProteinNew SeriesPharmaceutical ChemistryTumor Biology +15

Identification of the Spiro(oxindole-3,3′-thiazolidine)-Based Derivatives as Potential p53 Activity Modulators

Isabel Gómez‐Monterrey, Alessia Bertamino, Amalia Porta, +14

Journal of Medicinal Chemistry

Bioorganic ChemistryPharmacotherapyChemical BiologyPharmaceutical ChemistryRedox Biology +17

Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines

Marina Sala, Adele Chimento, Carmela Saturnino, +11

Bioorganic & Medicinal Chemistry Letters

Cytotoxic Activity EvaluationBiochemistryMedicine2,3-Thiazolidin-4-one DerivativesAnti-cancer Agent +3

2,6-Disubstituted imidazo[2,1-b][1,3,4]thiadiazole derivatives as potent staphylococcal biofilm inhibitors

Stella Cascioferro, Barbara Parrino, Giovanna Li Petri, +7

European Journal of Medicinal Chemistry

Medicinal ChemistryMedicineAntibacterial AgentMicrobiologyAntimicrobial Compound +2

New 1,2,4-Oxadiazole Nortopsentin Derivatives with Cytotoxic Activity

Stella Cascioferro, Alessandro Attanzio, Veronica Di Sarno, +5

Marine Drugs

1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A

Barbara Parrino, Daniela Carbone, Stella Cascioferro, +10

European Journal of Medicinal Chemistry

Staphylococcal Biofilm InhibitorsAntibioticsAntibacterial AgentMicrobiologyInfection Control +6

1,2,4‐Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase

Daniela Carbone, Barbara Parrino, Stella Cascioferro, +7

ChemMedChem

Biological activity of 3-chloro-azetidin-2-one derivatives having interesting antiproliferative activity on human breast cancer cell lines

Adele Chimento, Marina Sala, Isabel Gómez‐Monterrey, +13

Bioorganic & Medicinal Chemistry Letters

Biological ActivityBiochemistryMedicineNatural SciencesPharmacological Agent +4

Identification of a Potent Tryptophan-Based TRPM8 Antagonist With in Vivo Analgesic Activity

Alessia Bertamino, Nunzio Iraci, Carmine Ostacolo, +15

Journal of Medicinal Chemistry

Tryptamine-Based Derivatives as Transient Receptor Potential Melastatin Type 8 (TRPM8) Channel Modulators

Alessia Bertamino, Carmine Ostacolo, Paolo Ambrosino, +13

Journal of Medicinal Chemistry

Channel ModulatorsPain MedicineSynaptic TransmissionMolecular PainPharmacotherapy +23