Emiliano Rosatelli

Discovery of 6α-Ethyl-23(<i>S</i>)-methylcholic Acid (<i>S</i>-EMCA, INT-777) as a Potent and Selective Agonist for the TGR5 Receptor, a Novel Target for Diabesity

Roberto Pellicciari, Antimo Gioiello, Antonio Macchiarulo et al. · Journal of Medicinal Chemistry · 2009 · 255 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Building a Sulfonamide Library by Eco-Friendly Flow Synthesis

Antimo Gioiello, Emiliano Rosatelli, Michela Teofrasti et al. · ACS Combinatorial Science · 2013 · 71 citations

Pharmacy, Chemistry, Medicinal Chemistry +10

Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonists

Maura Marinozzi, Andrea Carotti, Emanuele Sansone et al. · Bioorganic & Medicinal Chemistry · 2012 · 44 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +9

Structure activity relationship of selective GABA uptake inhibitors

Stine B. Vogensen, Lars Jørgensen, Karsten K. Madsen et al. · Bioorganic & Medicinal Chemistry · 2015 · 31 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +14

Molecular Field Analysis and 3D-Quantitative Structure−Activity Relationship Study (MFA 3D-QSAR) Unveil Novel Features of Bile Acid Recognition at TGR5

Antonio Macchiarulo, Antimo Gioiello, Charles Thomas et al. · Journal of Chemical Information and Modeling · 2008 · 25 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17