Concepedia

Margaret Clackers

MC

Statistics

Publications

5

Citations

203

H-Index

5

Active since

2005

Affiliations

GlaxoSmithKline (United Kingdom)(Current)

GlaxoSmithKline (Ireland)

Margaret Clackers is an author at GlaxoSmithKline (United Kingdom) specializing in pharmacology, medicinal chemistry, and molecular pharmacology.

Publications per year

2005–2009

5

Publications

5

Dissociated Nonsteroidal Glucocorticoid Receptor Modulators; Discovery of the Agonist Trigger in a Tetrahydronaphthalene−Benzoxazine Series

Mike D. Barker, Margaret Clackers, Royston C. B. Copley et al. · Journal of Medicinal Chemistry · 2006 · 77 citations · Full text

, , +17

Design and Synthesis of New Nonsteroidal Glucocorticoid Modulators through Application of an “Agreement Docking” Method

Mike D. Barker, Margaret Clackers, Derek A. Demaine et al. · Journal of Medicinal Chemistry · 2005 · 44 citations · Full text

, , +17

Nonsteroidal Glucocorticoid Agonists: Tetrahydronaphthalenes with Alternative Steroidal A-Ring Mimetics Possessing Dissociated (Transrepression/Transactivation) Efficacy Selectivity

Keith Biggadike, Mohamed Boudjelal, Margaret Clackers et al. · Journal of Medicinal Chemistry · 2007 · 41 citations · Full text

, , +13

Non-steroidal glucocorticoid agonists—The discovery of aryl pyrazoles as A-ring mimetics

Margaret Clackers, Diane M. Coe, Derek A. Demaine et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 30 citations · Full text

, , +16

Highly tractable, sub-nanomolar non-steroidal glucocorticoid receptor agonists

Keith Biggadike, Matilde Caivano, Margaret Clackers et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 11 citations · Full text

, , +10

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