Cristina Gardelli

Discovery of Raltegravir, a Potent, Selective Orally Bioavailable HIV-Integrase Inhibitor for the Treatment of HIV-AIDS Infection

Vincenzo Summa, Alessia Petrocchi, Fabio Bonelli et al. · Journal of Medicinal Chemistry · 2008 · 634 citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +17

4,5-Dihydroxypyrimidine Carboxamides and <i>N</i>-Alkyl-5-hydroxypyrimidinone Carboxamides Are Potent, Selective HIV Integrase Inhibitors with Good Pharmacokinetic Profiles in Preclinical Species

Vincenzo Summa, Alessia Petrocchi, Victor G. Matassa et al. · Journal of Medicinal Chemistry · 2006 · 100 citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +13

Enantioselective Total Synthesis of the Antitumor Macrolide Rhizoxin D

Jennifer Lafontaine, David P. Provencal, Cristina Gardelli et al. · The Journal of Organic Chemistry · 2003 · 89 citations

Pharmacy, Chemistry, Medicinal Chemistry +9

Regiochemical control of the ring opening of 1,2-epoxides by means of chelating processes. 5. Synthesis and reactions of some 2,3-epoxy-1-alkanol derivatives

Marco Chini, Paolo Crotti, Lee A. Flippin et al. · The Journal of Organic Chemistry · 1993 · 89 citations

Natural Sciences, Biochemistry, Chemistry +7

Dihydroxypyrimidine-4-carboxamides as Novel Potent and Selective HIV Integrase Inhibitors

Paola Pace, Maria Emilia Di Francesco, Cristina Gardelli et al. · Journal of Medicinal Chemistry · 2007 · 77 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14