Serge Belanger

Potent, Orally Bioavailable Delta Opioid Receptor Agonists for the Treatment of Pain: Discovery of<i>N</i>,<i>N</i>-Diethyl-4-(5-hydroxyspiro[chromene-2,4′-piperidine]-4-yl)benzamide (ADL5859)

Bertrand Le Bourdonnec, Rolf T. Windh, Christopher W. Ajello et al. · Journal of Medicinal Chemistry · 2008 · 90 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Spirocyclic Delta Opioid Receptor Agonists for the Treatment of Pain: Discovery of<i>N</i>,<i>N</i>-Diethyl-3-hydroxy-4-(spiro[chromene-2,4′-piperidine]-4-yl) Benzamide (ADL5747)

Bertrand Le Bourdonnec, Rolf T. Windh, Lara K. Leister et al. · Journal of Medicinal Chemistry · 2009 · 85 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13

Expression of calcitonin gene-related peptide, substance P and protein kinase C in cultured dorsal root ganglion neurons following chronic exposure to mu, delta and kappa opiates

Serge Belanger, W Ma, J.‐G. Chabot et al. · Neuroscience · 2002 · 85 citations

Life Sciences, Neurobiology, Neuroscience +17

Novel malonamide derivatives as potent κ opioid receptor agonists

Guo‐Hua Chu, Minghua Gu, Joel Cassel et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 28 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +10

Elucidation of the Bioactive Conformation of the <i>N</i>-Substituted <i>trans</i>-3,4-Dimethyl-4-(3-hydroxyphenyl)piperidine Class of μ-Opioid Receptor Antagonists

Bertrand Le Bourdonnec, Mathieu Michaut, Hai‐Fen Ye et al. · Journal of Medicinal Chemistry · 2006 · 28 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17