Gary A. De Crescenzo

Solution structure and backbone dynamics of the catalytic domain of matrix metalloproteinase-2 complexed with a hydroxamic acid inhibitor

Yiqing Feng, John J. Likos, Leiming Zhu et al. · Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics · 2002 · 100 citations

Protein Chemistry, Catalytic Domain, Hydroxamic Acid Inhibitor +9

Discovery of novel benzothiazolesulfonamides as potent inhibitors of HIV-1 protease

Srinivasan Nagarajan, Gary A. De Crescenzo, Daniel P. Getman et al. · Bioorganic & Medicinal Chemistry · 2003 · 94 citations

Hiv-1 Protease, Biochemistry, Medicine +7

Synthesis and activity of selective MMP inhibitors with an aryl backbone

Thomas E. Barta, Daniel P. Becker, Louis J. Bedell et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 28 citations · Full text

Medicinal Chemistry, Selective Mmp Inhibitors, Biochemistry +8

Selective, orally active MMP inhibitors with an aryl backbone

Thomas E. Barta, Daniel P. Becker, Louis J. Bedell et al. · Bioorganic & Medicinal Chemistry Letters · 2001 · 17 citations · Full text

Medicinal Chemistry, Aryl Backbone, Medicine +6