Rui‐Yang Yang

Discovery and Optimization of a Series of 3-(3-Phenyl-3<i>H</i>-imidazo[4,5-<i>b</i>]pyridin-2-yl)pyridin-2-amines: Orally Bioavailable, Selective, and Potent ATP-Independent Akt Inhibitors

Mark A. Ashwell, Jean‐Marc Lapierre, Christopher J. Brassard et al. · Journal of Medicinal Chemistry · 2012 · 98 citations · Full text

Chemical Biology, Pharmaceutical Chemistry, Biophysical Screening Strategy +19

Solution and solid phase synthesis of 5-alkoxyhydantoin libraries with a three-fold functional diversity

Stephen Hanessian, Rui‐Yang Yang · Tetrahedron Letters · 1996 · 86 citations

Diversity Oriented Synthesis, Engineering, Organic Chemistry +6

The asymmetric synthesis of allylglycine and other unnatural α-amino acids via zinc-mediated allylation of oximes in aqueous media

Stephen Hanessian, Rui‐Yang Yang · Tetrahedron Letters · 1996 · 81 citations

Bioorganic Chemistry, Biochemistry, Natural Sciences +10

Synthetic methods for the preparation of ARQ 501 (β-Lapachone) human blood metabolites

Rui‐Yang Yang, Darin Kizer, Hui Wu et al. · Bioorganic & Medicinal Chemistry · 2008 · 58 citations

Biochemistry, Synthetic Methods, Medicine +7

A concise and efficient solid-phase synthesis of 2-amino-4(3H)-quinazolinones

Rui‐Yang Yang, Alan P. Kaplan · Tetrahedron Letters · 2000 · 51 citations

Organic Chemistry, Synthesis Method, Chemistry +2