Alan P. Kaplan

A concise and efficient solid-phase synthesis of 2-amino-4(3H)-quinazolinones

Rui‐Yang Yang, Alan P. Kaplan · Tetrahedron Letters · 2000 · 51 citations

Organic Chemistry, Synthesis Method, Chemistry +2

A new class of HIV-1 protease inhibitor: The crystallographic structure, inhibition and chemical synthesis of an aminimide peptide isostere

Earl Rutenber, Fiona McPhee, Alan P. Kaplan et al. · Bioorganic & Medicinal Chemistry · 1996 · 28 citations

Medicinal Chemistry, Hiv-1 Protease Inhibitor, Biochemistry +12

Reaction of isothiourea with 2,3-diaza-3-pentenedioic anhydride. A solid-phase synthesis of 3-amino-1,2,4-triazin-5(4H)-ones

Rui‐Yang Yang, Alan P. Kaplan · Tetrahedron Letters · 2001 · 19 citations

Solid-phase Synthesis, Engineering, Biochemistry +7

Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties

Vincent J. Santora, Theresa A. Almos, Richard Barido et al. · Journal of Medicinal Chemistry · 2018 · 18 citations · Full text

Pharmaceutical Science, Potent Glyt1 Inhibitors, Pharmacotherapy +16