Rajeshwar Singh

Discovery of a Novel Class of Boron-Based Antibacterials with Activity against Gram-Negative Bacteria

Vincent Hernandez, Thibaut Crépin, Andrés Palencia et al. · Antimicrobial Agents and Chemotherapy · 2013 · 195 citations · Full text

Available Antibiotics, Microbial Pathogens, Lead Analogue +24

Boron‐based phosphodiesterase inhibitors show novel binding of boron to PDE4 bimetal center

Yvonne R. Freund, Tsutomu Akama, M.R. Alley et al. · FEBS Letters · 2012 · 107 citations · Full text

Pharmaceutical Science, Phosphodiesterase 4, Pharmacotherapy +21

Identification of a novel boron-containing antibacterial agent (AN0128) with anti-inflammatory activity, for the potential treatment of cutaneous diseases

Stephen J. Baker, Tsutomu Akama, Yong-Kang Zhang et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 84 citations

Inflammation, Medicinal Chemistry, Anti-inflammatory +12

Synthesis and structural–activity relationships of 3-hydroxyquinazoline-2,4-dione antibacterial agents

Tuan P. Tran, Edmund L. Ellsworth, Michael A. Stier et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 75 citations

Antimicrobial Drug Discovery, Medicine, Antibacterial Agent +3

First and Second Generation γ-Secretase Modulators (GSMs) Modulate Amyloid-β (Aβ) Peptide Production through Different Mechanisms

Tomas Borgegård, Anders Juréus, Fredrik Olsson et al. · Journal of Biological Chemistry · 2012 · 74 citations · Full text