Graham G. A. Inglis

Expanding GSK's solvent selection guide – embedding sustainability into solvent selection starting at medicinal chemistry

Richard K. Henderson, Concepción Jiménez‐González, David J. C. Constable et al. · Green Chemistry · 2011 · 1.1K citations

Pharmaceutical Science, Pharmaceutical Research, Engineering +23

An Extremely Powerful Acylation Reaction of Alcohols with Acid Anhydrides Catalyzed by Trimethylsilyl Trifluoromethanesulfonate

Panayiotis A. Procopiou, Simon P. D. Baugh, Stephen S. Flack et al. · The Journal of Organic Chemistry · 1998 · 258 citations

Standard Dmap Conditions, Cross-coupling Reaction, Engineering +13

An extremely fast and efficient acylation reaction of alcohols with acid anhydrides in the presence of trimethylsilyl trifluoromethanesulfonate as catalyst

Panayiotis A. Procopiou, Simon P. D. Baugh, Stephen S. Flack et al. · Chemical Communications · 1996 · 88 citations

Engineering, Organic Chemistry, Acid Anhydrides +20

Dimeric Zanamivir Conjugates with Various Linking Groups Are Potent, Long-Lasting Inhibitors of Influenza Neuraminidase Including H5N1 Avian Influenza

Simon J. F. Macdonald, Rachel Cameron, Derek A. Demaine et al. · Journal of Medicinal Chemistry · 2005 · 87 citations · Full text

Medicinal Chemistry, Medicine, Plaque Reduction Assays +14

Potent and Long-Acting Dimeric Inhibitors of Influenza Virus Neuraminidase Are Effective at a Once-Weekly Dosing Regimen

Simon J. F. Macdonald, Keith G. Watson, Rachel Cameron et al. · Antimicrobial Agents and Chemotherapy · 2004 · 80 citations · Full text

Medicinal Chemistry, Antiviral Compound, Medicine +12