Roberto Rigolio

Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 1. Identification of the 4-Quinolinecarboxamide Framework

Giuseppe Giardina, Henry M. Sarau, Carlo Farina et al. · Journal of Medicinal Chemistry · 1997 · 79 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (<i>S</i>)-<i>N</i>-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)

Giuseppe Giardina, Luca F. Raveglia, Mario Grugni et al. · Journal of Medicinal Chemistry · 1999 · 63 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +14

2-Phenyl-4-quinolinecarboxamides:  A Novel Class of Potent and Selective Non-Peptide Competitive Antagonists for the Human Neurokinin-3 Receptor

Giuseppe Giardina, Henry M. Sarau, Carlo Farina et al. · Journal of Medicinal Chemistry · 1996 · 47 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +7

Replacement of the quinoline system in 2-phenyl-4-quinolinecarboxamide NK-3 receptor antagonists

Giuseppe Giardina, Marco Artico, Stefano Cavagnera et al. · Il Farmaco · 1999 · 21 citations

Medicine, Medicinal Chemistry, Pharmacology +11

A reliable and efficient synthesis of SR 142801

Giuseppe Giardina, Mario Grugni, Roberto Rigolio et al. · Bioorganic & Medicinal Chemistry Letters · 1996 · 17 citations

Natural Sciences, Chemistry, Materials Science +2