Concepedia

Mario Grugni

MG

Statistics

Publications

13

Citations

500

H-Index

12

Active since

1995

Affiliations

New Frontier(Current)

CTI BioPharma (United Kingdom)

Mario Grugni is an author at New Frontier specializing in medicinal chemistry, pharmacology, and neuropharmacology.

Publications per year

1995–2010

13

Publications

13

Nonpeptide Tachykinin Receptor Antagonists. III. SB 235375, a Low Central Nervous System-Penetrant, Potent and Selective Neurokinin-3 Receptor Antagonist, Inhibits Citric Acid-Induced Cough and Airways Hyper-reactivity in Guinea Pigs

Douglas W.P. Hay, Giuseppe Giardina, Don E. Griswold et al. · Journal of Pharmacology and Experimental Therapeutics · 2002 · 90 citations · Full text

, , +13

Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 1. Identification of the 4-Quinolinecarboxamide Framework

Giuseppe Giardina, Henry M. Sarau, Carlo Farina et al. · Journal of Medicinal Chemistry · 1997 · 79 citations · Full text

, , +12

Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (<i>S</i>)-<i>N</i>-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)

Giuseppe Giardina, Luca F. Raveglia, Mario Grugni et al. · Journal of Medicinal Chemistry · 1999 · 63 citations · Full text

, , +14

2-Phenyl-4-quinolinecarboxamides:  A Novel Class of Potent and Selective Non-Peptide Competitive Antagonists for the Human Neurokinin-3 Receptor

Giuseppe Giardina, Henry M. Sarau, Carlo Farina et al. · Journal of Medicinal Chemistry · 1996 · 47 citations · Full text

, , +7

Stepwise Modulation of Neurokinin-3 and Neurokinin-2 Receptor Affinity and Selectivity in Quinoline Tachykinin Receptor Antagonists

Frank E. Blaney, Luca F. Raveglia, Marco Artico et al. · Journal of Medicinal Chemistry · 2001 · 45 citations · Full text

, , +16

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