Discovery of a Novel Antitumor Benzolactone Enamide Class That Selectively Inhibits Mammalian Vacuolar-Type (H+)-ATPases

Michael R. Boyd, Carlo Farina, Pietro Belfiore, +6

Journal of Pharmacology and Experimental Therapeutics

A selective inhibitor of the osteoclastic V-H+-ATPase prevents bone loss in both thyroparathyroidectomized and ovariectomized rats

L. Visentin, Robert A. Dodds, Maurizio Valente, +6

Journal of Clinical Investigation

Percutaneous transluminal angioplasty versus surgery for subclavian artery occlusive disease

Carlo Farina, Andrea Mingoli, Richard D. Schultz, +4

The American Journal of Surgery

Endovascular TechniqueVascular SurgeryThoracic SurgerySurgeryEndovascular Management +2

Elevated levels of a C-terminal agrin fragment identifies a new subset of sarcopenia patients

Stefan Hettwer, Pius Dahinden, Stefan Kucsera, +6

Experimental Gerontology

C-terminal Agrin FragmentClinical PhysiologyElevated LevelsClinical InjurySarcopenia +12

Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 1. Identification of the 4-Quinolinecarboxamide Framework

Giuseppe Giardina, Henry M. Sarau, Carlo Farina, +8

Journal of Medicinal Chemistry

4-Quinolinecarboxamide FrameworkReceptor AntagonistsPharmacotherapyPharmaceutical ChemistryMembrane Preparation +16

Long-term outcome after transaxillary approach for thoracic outlet syndrome

Andrea Mingoli, Richard J. Feldhaus, Carlo Farina, +4

Surgery

Spinal Cord InjuryTransaxillary ApproachThoracic SurgerySurgeryThoracic Spine +2

5-(5,6-Dichloro-2-indolyl)-2-methoxy-2,4-pentadienamides:  Novel and Selective Inhibitors of the Vacuolar H⁺-ATPase of Osteoclasts with Bone Antiresorptive Activity

Stefania Gagliardi, Guy Nadler, Emanuela Consolandi, +10

Journal of Medicinal Chemistry

Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (<i>S</i>)-<i>N</i>-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)

Giuseppe Giardina, Luca F. Raveglia, Mario Grugni, +11

Journal of Medicinal Chemistry

Position 3Peptide SciencePharmacotherapyChemical BiologyMolecular Pharmacology +16

Synthesis and Structure−Activity Relationships of Bafilomycin A₁ Derivatives as Inhibitors of Vacuolar H⁺-ATPase

Stefania Gagliardi, Pier Andrea Gatti, Pietro Belfiore, +3

Journal of Medicinal Chemistry

Molecular PharmacologyMedicinal ChemistryBafilomycin A1Bioorganic ChemistryBiochemistry +12

Discovery of a Novel Class of Substituted Pyrrolooctahydroisoquinolines as Potent and Selective δ Opioid Agonists, Based on an Extension of the Message−Address Concept

Giulio Dondio, Silvano Ronzoni, Drake S. Eggleston, +7

Journal of Medicinal Chemistry