A reliable and efficient synthesis of SR 142801

Selective Removal of the Tert-Butoxycarbonyl Group from Secondary Amines: ZnBr₂as the Deprotecting Reagent

Satish C. Nigama, André Mann, Maurizio Taddei et al. · Synthetic Communications · 1989 · 64 citations

Natural Sciences, Chemistry, Organic Chemistry +6

Functional characterization of the nonpeptide neurokinin3 (NK3) receptor antagonist, SR142801 on the human NK3 receptor expressed in Chinese hamster ovary cells.

Florence Oury-Donat, P Carayon, O. Thurneyssen et al. · Journal of Pharmacology and Experimental Therapeutics · 1995 · 58 citations · Full text

Medicine, Pharmacology, Molecular Pharmacology +8

2-Phenyl-4-quinolinecarboxamides:  A Novel Class of Potent and Selective Non-Peptide Competitive Antagonists for the Human Neurokinin-3 Receptor

Giuseppe Giardina, Henry M. Sarau, Carlo Farina et al. · Journal of Medicinal Chemistry · 1996 · 47 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +7

The development of a novel series of non-peptide tachykinin NK3 receptor selective antagonists

P. Boden, J.M. Eden, Julie Hodgson et al. · Bioorganic & Medicinal Chemistry Letters · 1995 · 28 citations

Medicine, Medicinal Chemistry, Pharmacology +8

Über Alkylenimin‐Derivate. 2. Mitteilung

E. Tagmann, E. Sury, K. Hoffmann · Helvetica Chimica Acta · 1952 · 27 citations

Medicine, Medicinal Chemistry, Pharmacology +8