Matthew Whiting

Inhibitors of HIV‐1 Protease by Using In Situ Click Chemistry

Matthew Whiting, John Muldoon, Ying‐Chuan Lin et al. · Angewandte Chemie International Edition · 2006 · 506 citations

Poor Equals Potent, Click Chemistry, Antiviral Drug +17

Rapid Discovery and Structure−Activity Profiling of Novel Inhibitors of Human Immunodeficiency Virus Type 1 Protease Enabled by the Copper(I)-Catalyzed Synthesis of 1,2,3-Triazoles and Their Further Functionalization

Matthew Whiting, Jonathan C. Tripp, Ying‐Chuan Lin et al. · Journal of Medicinal Chemistry · 2006 · 206 citations · Full text

Combinatorial Chemistry, Structure−activity Profiling, Click Chemistry +16

Copper‐Catalyzed Reaction Cascade: Direct Conversion of Alkynes into <i>N</i>‐Sulfonylazetidin‐2‐imines

Matthew Whiting, Valery V. Fokin · Angewandte Chemie International Edition · 2006 · 166 citations

Asymmetric Catalysis, Cross-coupling Reaction, Engineering +10

Potential for the Formation of <i>N</i>-Nitrosamines during the Manufacture of Active Pharmaceutical Ingredients: An Assessment of the Risk Posed by Trace Nitrite in Water

Ian W. Ashworth, Olivier Dirat, Andrew Teasdale et al. · Organic Process Research & Development · 2020 · 119 citations

Pharmaceutical Science, Engineering, Chemical Analysis +22

Inhibitors of HIV‐1 Protease by Using In Situ Click Chemistry

Matthew Whiting, John Muldoon, Ying‐Chuan Lin et al. · Angewandte Chemie · 2006 · 89 citations

Die Triazolverknüpfung Erzeugt, Immunology, Pharmacotherapy +19