Etienne J. Donckèle

An ultra-high-affinity small organic ligand of fibroblast activation protein for tumor-targeting applications

Jacopo Millul, Gabriele Bassi, Jacqueline Mock et al. · Proceedings of the National Academy of Sciences · 2021 · 145 citations · Full text

Palladium‐Catalyzed Enantioselective Allylic Alkylations through C–H Activation

Barry M. Trost, David A. Thaisrivongs, Etienne J. Donckèle · Angewandte Chemie International Edition · 2012 · 140 citations

Medicinal Chemistry, Enantioselective Synthesis, Engineering +12

Synthesis and Profiling of a Diverse Collection of Azetidine-Based Scaffolds for the Development of CNS-Focused Lead-like Libraries

Jason T. Lowe, Maurice D. Lee, Lakshmi B. Akella et al. · The Journal of Organic Chemistry · 2012 · 135 citations · Full text

Combinatorial Chemistry, Bioorganic Chemistry, Lead Identification +18

A New Class of Non-<i>C</i>₂-Symmetric Ligands for Oxidative and Redox-Neutral Palladium-Catalyzed Asymmetric Allylic Alkylations of 1,3-Diketones

Barry M. Trost, Etienne J. Donckèle, David A. Thaisrivongs et al. · Journal of the American Chemical Society · 2015 · 98 citations · Full text

Cross-coupling Reaction, Chiral Products, Engineering +10

Enantioselective Catalysis Coupled with Stereodivergent Cyclization Strategies Enables Rapid Syntheses of (+)‐Limaspermidine and (+)‐Kopsihainanine A

Beau P. Pritchett, Etienne J. Donckèle, Brian M. Stoltz · Angewandte Chemie International Edition · 2017 · 66 citations · Full text