George Derbin

Discovery of Brivanib Alaninate ((<i>S</i>)-((<i>R</i>)-1-(4-(4-Fluoro-2-methyl-1<i>H</i>-indol-5-yloxy)-5-methylpyrrolo[2,1-<i>f</i>][1,2,4]triazin-6-yloxy)propan-2-yl)2-aminopropanoate), A Novel Prodrug of Dual Vascular Endothelial Growth Factor Receptor-2 and Fibroblast Growth Factor Receptor-1 Kinase Inhibitor (BMS-540215)

Zhen‐Wei Cai, Yongzheng Zhang, R. M. Borzilleri et al. · Journal of Medicinal Chemistry · 2008 · 141 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Discovery and Preclinical Studies of (<i>R</i>)-1-(4-(4-Fluoro-2-methyl-1<i>H</i>-indol-5-yloxy)-5- methylpyrrolo[2,1-<i>f</i>][1,2,4]triazin-6-yloxy)propan- 2-ol (BMS-540215), an In Vivo Active Potent VEGFR-2 Inhibitor

Rajeev S. Bhide, Zhen‐Wei Cai, Yong‐Zheng Zhang et al. · Journal of Medicinal Chemistry · 2006 · 133 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Discovery and Evaluation of <i>N</i>-Cyclopropyl- 2,4-difluoro-5-((2-(pyridin-2-ylamino)thiazol-5- ylmethyl)amino)benzamide (BMS-605541), a Selective and Orally Efficacious Inhibitor of Vascular Endothelial Growth Factor Receptor-2

R. M. Borzilleri, Rajeev S. Bhide, Joel C. Barrish et al. · Journal of Medicinal Chemistry · 2006 · 40 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Development of a Canine Model to Enable the Preclinical Assessment of Ph-dependent Absorption of Test Compounds

R. Marcus Fancher, Hongjian Zhang, Bogdan Sleczka et al. · Journal of Pharmaceutical Sciences · 2011 · 30 citations

Pharmacy, Pharmacokinetics, Pharmacology +13

Circumvention of pH-dependent release from ethylcellulosecoated pellets

J.B. Dressman, George Derbin, George Ismailos et al. · Journal of Controlled Release · 1995 · 21 citations

Pharmacy, Pharmaceutics, Dissolution Testing +7