Graham F. Joiner

5-Chloro-<i>N</i>-(4-methoxy-3-piperazin-1-yl- phenyl)-3-methyl-2-benzothiophenesulfon- amide (SB-271046):  A Potent, Selective, and Orally Bioavailable 5-HT₆ Receptor Antagonist

Steven M. Bromidge, Anthony M. Brown, Stephen E. Clarke et al. · Journal of Medicinal Chemistry · 1999 · 170 citations · Full text

Drug Target, Altmetric Attention Score, 4-Methoxy-3-piperazin-1-yl- Phenyl +18

5-Hydroxytryptamine (5-HT3) receptor antagonists. 1. Indazole and indolizine-3-carboxylic acid derivatives

José Luis Bermúdez, Charles S. Fake, Graham F. Joiner et al. · Journal of Medicinal Chemistry · 1990 · 152 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Conformational Restriction +14

The Selective 5-HT_1BReceptor Inverse Agonist 1‘-Methyl-5-[[2‘-methyl-4‘- (5-methyl-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl]-2,3,6,7-tetrahydro- spiro[furo[2,3-<i>f</i>]indole-3,4‘-piperidine] (SB-224289) Potently Blocks Terminal 5-HT Autoreceptor Function Both in Vitro and in Vivo

Laramie M. Gaster, Frank E. Blaney, Susannah Davies et al. · Journal of Medicinal Chemistry · 1998 · 81 citations · Full text

Phenyl benzenesulfonamides are novel and selective 5-HT6 antagonists: identification of N-(2,5-dibromo-3-fluorophenyl)-4-methoxy-3-piperazin-1-ylbenzenesulfonamide (SB-357134)

Steven M. Bromidge, Stephen E. Clarke, Tracey Gager et al. · Bioorganic & Medicinal Chemistry Letters · 2001 · 56 citations · Full text

Selective 5-Ht6 Antagonists, Medicinal Chemistry, Derivative (Chemistry) +10

N-[(1-Butyl-4-piperidinyl)methyl]-3,4- dihydro-2H-[1,3]oxazino[3,2-a]indole- 10-carboxamide hydrochloride: the first potent and selective 5-HT4 receptor antagonist amide with oral activity.

Laramie M. Gaster, Graham F. Joiner, F. D. KING et al. · Journal of Medicinal Chemistry · 1995 · 43 citations · Full text

Pharmaceutical Science, Altmetric Attention Score, Organic Chemistry +19