Concepedia
Statistics
Publications
8
Citations
260
H-Index
Active since
2017
Affiliations
Goethe University Frankfurt(Current)
Fraunhofer Institute for Molecular Biology and Applied Ecology
Fraunhofer Institute for Translational Medicine and Pharmacology
Leonie Gellrich is an author at Goethe University Frankfurt specializing in pharmacology, medicinal chemistry, and drug discovery.
Publications per year
2017–2021
Tuning Nuclear Receptor Selectivity of Wy14,643 towards Selective Retinoid X Receptor Modulation
Julius Pollinger, Leonie Gellrich, Simone Schierle et al. · Journal of Medicinal Chemistry · 2019 · 54 citations · Full text
Medicine, Medicinal Chemistry, Pharmacology +16
Endogenous vitamin E metabolites mediate allosteric PPARγ activation with unprecedented co-regulatory interactions
Sabine Willems, Leonie Gellrich, A. Chaikuad et al. · Cell chemical biology · 2021 · 53 citations
Life Sciences, Biochemistry, Pharmacology +16
<scp>l</scp>-Thyroxin and the Nonclassical Thyroid Hormone TETRAC Are Potent Activators of PPARγ
Leonie Gellrich, Pascal Heitel, Jan Heering et al. · Journal of Medicinal Chemistry · 2020 · 49 citations · Full text
Life Sciences, Biochemistry, Pharmacology +17
Computer-Assisted Discovery and Structural Optimization of a Novel Retinoid X Receptor Agonist Chemotype
Pascal Heitel, Leonie Gellrich, Lena Kalinowsky et al. · ACS Medicinal Chemistry Letters · 2019 · 45 citations · Full text
Pharmacy, Medicinal Chemistry, Pharmacology +17
Urate transporter inhibitor lesinurad is a selective peroxisome proliferator-activated receptor gamma modulator (sPPARγM) in vitro
Pascal Heitel, Leonie Gellrich, Jan Heering et al. · Scientific Reports · 2018 · 21 citations · Full text
Medicine, Medicinal Chemistry, Pharmacology +14
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