Thomas Drapier

Enhancing Action of Positive Allosteric Modulators through the Design of Dimeric Compounds

Thomas Drapier, Pierre Geubelle, Charlotte Bouckaert et al. · Journal of Medicinal Chemistry · 2018 · 48 citations · Full text

7-Phenoxy-Substituted 3,4-Dihydro-2<i>H</i>-1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar Potency

Eric Goffin, Thomas Drapier, A.P. Larsen et al. · Journal of Medicinal Chemistry · 2017 · 45 citations · Full text

Crystal Structures of Potent Dimeric Positive Allosteric Modulators at the Ligand-Binding Domain of the GluA2 Receptor

Saara Laulumaa, Kathrine Voigt Hansen, Magdalena Masternak et al. · ACS Medicinal Chemistry Letters · 2018 · 10 citations