Pierre Geubelle

Identification and pharmacological characterization of succinate receptor agonists

Pierre Geubelle, Julie Gilissen, Sébastien Dilly et al. · British Journal of Pharmacology · 2017 · 62 citations · Full text

Forskolin-free cAMP assay for Gi-coupled receptors

Julie Gilissen, Pierre Geubelle, Nadine Dupuis et al. · Biochemical Pharmacology · 2015 · 50 citations

Signal Transduction, G Protein-coupled Receptor, Medicine +5

Enhancing Action of Positive Allosteric Modulators through the Design of Dimeric Compounds

Thomas Drapier, Pierre Geubelle, Charlotte Bouckaert et al. · Journal of Medicinal Chemistry · 2018 · 48 citations · Full text

7-Phenoxy-Substituted 3,4-Dihydro-2<i>H</i>-1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar Potency

Eric Goffin, Thomas Drapier, A.P. Larsen et al. · Journal of Medicinal Chemistry · 2017 · 45 citations · Full text

Activation of the Orphan G Protein–Coupled Receptor GPR27 by Surrogate Ligands Promotes β-Arrestin 2 Recruitment

Nadine Dupuis, Céline Laschet, Delphine Franssen et al. · Molecular Pharmacology · 2017 · 34 citations · Full text