Helen J. Mason

Parallel Synthesis of Aldehydes and Ketone Facilitated by a New Solid-Phase Weinreb Amide

Joseph M. Salvino, Miljenko Mervič, Helen J. Mason et al. · The Journal of Organic Chemistry · 1999 · 49 citations

Combinatorial Chemistry, Engineering, Organic Chemistry +16

Substituted Pyrazolopyridines as Potent and Selective PDE5 Inhibitors:  Potential Agents for Treatment of Erectile Dysfunction

Guixue Yu, Helen J. Mason, Ximao Wu et al. · Journal of Medicinal Chemistry · 2001 · 45 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Urology +14

Design and Structure−Activity Relationships of Potent and Selective Inhibitors of Blood Coagulation Factor Xa

William R. Ewing, Michael R. Becker, Vincent E. Manetta et al. · Journal of Medicinal Chemistry · 1999 · 42 citations · Full text

Selective Inhibitors, Pharmacotherapy, Chemical Biology +19

An Imidazopiperidine Series of CCR5 Antagonists for the Treatment of HIV: The Discovery of <i>N</i>-{(1<i>S</i>)-1-(3-Fluorophenyl)-3-[(3-<i>endo</i>)-3-(5-isobutyryl-2-methyl-4,5,6,7-tetrahydro-1<i>H</i>-imidazo[4,5-<i>c</i>]pyridin-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]propyl}acetamide (PF-232798)

Paul A. Stupple, David V. Batchelor, Martin Corless et al. · Journal of Medicinal Chemistry · 2010 · 40 citations · Full text

Medicinal Chemistry, Maraviroc 1, Imidazopiperidine Series +15

Sulfonamidopyrrolidinone Factor Xa Inhibitors:  Potency and Selectivity Enhancements via P-1 and P-4 Optimization

Yong Mi Choi-Sledeski, Daniel McGarry, Daniel M. Green et al. · Journal of Medicinal Chemistry · 1999 · 36 citations · Full text

Pharmaceutical Science, Bioorganic Chemistry, Pharmacotherapy +18