Tobias Grabe

Inhibition of osimertinib-resistant epidermal growth factor receptor EGFR-T790M/C797S

Jonas Lategahn, Marina Keul, Philip Klövekorn et al. · Chemical Science · 2019 · 52 citations · Full text

Medicine, Oncology, Pharmacology +16

Complex Crystal Structures of EGFR with Third-Generation Kinase Inhibitors and Simultaneously Bound Allosteric Ligands

Janina Niggenaber, Leonie Heyden, Tobias Grabe et al. · ACS Medicinal Chemistry Letters · 2020 · 51 citations · Full text

Medicine, Medicinal Chemistry, Oncology +13

Synthesis of well-defined core–shell nanoparticles based on bifunctional poly(2-oxazoline) macromonomer surfactants and a microemulsion polymerization process

Anne‐Larissa Kampmann, Tobias Grabe, Carolin Jaworski et al. · RSC Advances · 2016 · 27 citations

Natural Sciences, Chemistry, Materials Science +17

Insight into Targeting Exon20 Insertion Mutations of the Epidermal Growth Factor Receptor with Wild Type-Sparing Inhibitors

Jonas Lategahn, Hannah L. Tumbrink, Carsten Schultz‐Fademrecht et al. · Journal of Medicinal Chemistry · 2022 · 23 citations

Medicine, Oncology, Pharmacology +14

Targeting Her2-insYVMA with Covalent Inhibitors—A Focused Compound Screening and Structure-Based Design Approach

Jonas Lategahn, Julia Hardick, Tobias Grabe et al. · Journal of Medicinal Chemistry · 2020 · 19 citations · Full text

Pharmacy, Medicinal Chemistry, Oncology +15