Jian Sun

Aminoethylenes:  A Tetrahedral Intermediate Isostere Yielding Potent Inhibitors of the Aspartyl Protease BACE-1

Wenjin Yang, Wanli Lu, Yafan Lu et al. · Journal of Medicinal Chemistry · 2006 · 52 citations · Full text

Fragment-Based Discovery of Nonpeptidic BACE-1 Inhibitors Using Tethering

Wenjin Yang, Raymond V. Fucini, Bruce J. Fahr et al. · Biochemistry · 2009 · 48 citations

Drug Target, Protein Assembly, Molecular Biology +18

Stereoselective Total Synthesis of Epothilones by the Metathesis Approach Involving C9−C10 Bond Formation

Jian Sun, Subhash C. Sinha · Angewandte Chemie International Edition · 2002 · 44 citations

A P(V)–N Activation Strategy for the Synthesis of Nucleoside Polyphosphates

Qi Sun, Shan‐Shan Gong, Jian Sun et al. · The Journal of Organic Chemistry · 2013 · 40 citations

Biosynthesis, P Nmr, Engineering +9

Sets of Aldolase Antibodies with Antipodal Reactivities. Formal Synthesis of Epothilone E by Large-Scale Antibody-Catalyzed Resolution of Thiazole Aldol

Subhash C. Sinha, Jian Sun, Carlos F. Barbas et al. · Organic Letters · 1999 · 40 citations

Diversity Oriented Synthesis, Bioorganic Chemistry, Antipodal Reactivities +15