Bruce L. Jacobson

Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP)

Richard Sulsky, David R. Magnin, Yanting Huang et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 150 citations · Full text

Lipid Synthesis, Biochemistry, Natural Sciences +6

Discovery of a 1<i>H</i>-Benzoimidazol-2-yl)-1<i>H</i>-pyridin-2-one (BMS-536924) Inhibitor of Insulin-like Growth Factor I Receptor Kinase with in Vivo Antitumor Activity

Mark D. Wittman, Joan M. Carboni, Ricardo M. Attar et al. · Journal of Medicinal Chemistry · 2005 · 134 citations · Full text

Pharmacotherapy, Insulin Receptor, Insulin Signaling +21

Sulfate-binding protein dislikes protonated oxyacids

Bruce L. Jacobson, Florante A. Quiocho · Journal of Molecular Biology · 1988 · 118 citations

Sulfate-binding Protein Dislikes, Structure-function Enzyme Kinetics, Protein Chemistry +1

Molecular structure of the oxidized, recombinant, heterocyst [2Fe-2S] (iron-sulfur) ferredoxin from Anabaena 7120 determined to 1.7-.ANG. resolution

Bruce L. Jacobson, Young Kee Chae, John L. Markley et al. · Biochemistry · 1993 · 86 citations

Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors

James Sutton, Scott A. Bolton, Malcolm E. Davis et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 63 citations · Full text

Medicinal Chemistry, Solid-phase Synthesis, Medicine +5