Tiziana Ginex

Identification of Dihydrofuro[3,4-<i>d</i>]pyrimidine Derivatives as Novel HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors with Promising Antiviral Activities and Desirable Physicochemical Properties

Dongwei Kang, Heng Zhang, Zhao Wang et al. · Journal of Medicinal Chemistry · 2019 · 86 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Combined in Vitro Cell-Based/in Silico Screening of Naturally Occurring Flavonoids and Phenolic Compounds as Potential Anti-Alzheimer Drugs

Alba Espargaró, Tiziana Ginex, Maria del Mar Vadell et al. · Journal of Natural Products · 2017 · 82 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Design, synthesis and docking study of novel coumarin ligands as potential selective acetylcholinesterase inhibitors

Fatih Sönmez, Belma Zengin Kurt, Livia Basile et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 2017 · 78 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Exploiting the Tolerant Region I of the Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI) Binding Pocket: Discovery of Potent Diarylpyrimidine-Typed HIV-1 NNRTIs against Wild-Type and E138K Mutant Virus with Significantly Improved Water Solubility and Favorable Safety Profiles

Boshi Huang, Wen‐Ming Chen, Tong Zhao et al. · Journal of Medicinal Chemistry · 2019 · 77 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Exploring the hydrophobic channel of NNIBP leads to the discovery of novel piperidine-substituted thiophene[3,2-d]pyrimidine derivatives as potent HIV-1 NNRTIs

Dongwei Kang, Da Feng, Tiziana Ginex et al. · Acta Pharmaceutica Sinica B · 2019 · 51 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17