Diego Dal Ben

Fragment optimization for GPCRs by molecular dynamics free energy calculations: Probing druggable subpockets of the A 2A adenosine receptor binding site

Pierre Matricon, Anirudh Ranganathan, Eugene Warnick et al. · Scientific Reports · 2017 · 64 citations · Full text

Design, synthesis and evaluation in an LPS rodent model of neuroinflammation of a novel 18F-labelled PET tracer targeting P2X7

E. Fantoni, Diego Dal Ben, Simonetta Falzoni et al. · EJNMMI Research · 2017 · 57 citations · Full text

Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17

Michela Buccioni, Gabriella Marucci, Diego Dal Ben et al. · Purinergic Signalling · 2011 · 56 citations · Full text

Molecular Pharmacology, Pharmacological Characterization, Signal Transduction +10

8-Bromo-9-alkyl adenine derivatives as tools for developing new adenosine A2A and A2B receptors ligands

Catia Lambertucci, Ippolito Antonini, Michela Buccioni et al. · Bioorganic & Medicinal Chemistry · 2009 · 55 citations · Full text

A2b Receptors Ligands, Biochemistry, G Protein-coupled Receptor +9

Pyrazolo[1,5-c]quinazoline derivatives and their simplified analogues as adenosine receptor antagonists: Synthesis, structure–affinity relationships and molecular modeling studies

Daniela Catarzi, Vittoria Colotta, Flavia Varano et al. · Bioorganic & Medicinal Chemistry · 2012 · 54 citations · Full text

Molecular Pharmacology, Biochemistry, Simplified Analogues +9