Anita Tertre

Crystal Structures of Novel Non-peptidic, Non-zinc Chelating Inhibitors Bound to MMP-12

Renaud Morales, Sophie Perrier, Jean-Michel Florent et al. · Journal of Molecular Biology · 2004 · 86 citations

Natural Sciences, Chemistry, Medicinal Chemistry +12

Structure-based design and synthesis of novel non-zinc chelating MMP-12 inhibitors

Anne‐Claude Dublanchet, Pierre Ducrot, Charles R. Andrianjara et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 69 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +14

Discovery of thiadiazoles as a novel structural class of potent and selective PDE7 inhibitors. Part 1: Design, synthesis and structure–activity relationship studies

Fabrice Vergne, Patrick Bernardelli, Edwige Lorthiois et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 57 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 1

Edwige Lorthiois, Patrick Bernardelli, Fabrice Vergne et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 50 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +7

Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 2: Optimization of 5,8-disubstituted derivatives

Patrick Bernardelli, Edwige Lorthiois, Fabrice Vergne et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 38 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12