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Structure-based design and synthesis of novel non-zinc chelating MMP-12 inhibitors

Anne‐Claude Dublanchet, Pierre Ducrot, Charles R. Andrianjara, Margaret O’Gara, Renaud Morales, Delphine Compère, Alexis Denis, Stéphane Blais, Philippe Cluzeau, Karine Courté,

Bioorganic & Medicinal Chemistry Letters · 2005 · 69 citations · 8 references

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8

Requirement for Macrophage Elastase for Cigarette Smoke-Induced Emphysema in Mice

R. Dean Hautamaki, Dale K. Kobayashi, Robert M. Senior et al. · Science · 1997 · 1.5K citations

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Crystal Engineering for Topochemical Polymerization of Muconic Esters Using Halogen−Halogen and CH/π Interactions as Weak Intermolecular Interactions

Akikazu Matsumoto, Toshihiro Tanaka, Takashi Tsubouchi et al. · Journal of the American Chemical Society · 2002 · 180 citations

, , +17

Matrix metalloproteinase inhibitors 1998

R. Paul Beckett, Mark Whittaker · Expert Opinion on Therapeutic Patents · 1998 · 133 citations

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Structure-Based Design of a Novel, Potent, and Selective Inhibitor for MMP-13 Utilizing NMR Spectroscopy and Computer-Aided Molecular Design

James Chen, Frances C. Nelson, Jeremy I. Levin et al. · Journal of the American Chemical Society · 2000 · 107 citations

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Substrate specificity determinants of human macrophage elastase (MMP-12) based on the 1.1 Å crystal structure 1 1Edited by I. Wilson

Andreas Kocourek, Marianne Braun, Harald Tschesche et al. · Journal of Molecular Biology · 2001 · 100 citations

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