Patrice Désos

S32826, A Nanomolar Inhibitor of Autotaxin: Discovery, Synthesis and Applications as a Pharmacological Tool

Gilles Ferry, Natacha Moulharat, Jean‐Philippe Pradère et al. · Journal of Pharmacology and Experimental Therapeutics · 2008 · 95 citations

Structure−Activity Relationships in a Series of 2(1<i>H</i>)-Quinolones Bearing Different Acidic Function in the 3-Position:  6,7-Dichloro-2(1<i>H</i>)-oxoquinoline-3-phosphonic Acid, a New Potent and Selective AMPA/Kainate Antagonist with Neuroprotective Properties

Patrice Désos, J. Lépagnol, Philippe Morain et al. · Journal of Medicinal Chemistry · 1996 · 77 citations

Enantioselective synthesis of a pyrrolo-benzothiadiazine derivative S 18986, a new AMPA receptor positive modulator

Patrice Désos, Bernard Serkiz, Philippe Morain et al. · Bioorganic & Medicinal Chemistry Letters · 1996 · 40 citations

Medicine, Organic Chemistry, Stereoselective Synthesis +5

Asymmetric Synthesis. 39.¹ Synthesis of 2-(1-Aminoalkyl)piperidines <i>via</i> 2-Cyano-6-phenyl Oxazolopiperidine

Olivier Froelich, Patrice Désos, Martine Bonin et al. · The Journal of Organic Chemistry · 1996 · 37 citations · Full text

Amine 19, Heterocyclic, Asymmetric Synthesis +6

DRUG FOCUS: S 18986: A Positive Allosteric Modulator of AMPA‐Type Glutamate Receptors Pharmacological Profile of a Novel Cognitive Enhancer

Katy Bernard, Laurence Danober, Jean‐Yves Thomas et al. · CNS Neuroscience & Therapeutics · 2010 · 35 citations · Full text

Novel Cognitive Enhancer, Synaptic Transmission, Neurotransmitter +19