Lutz Preu

10-Iodo-11<i>H</i>-indolo[3,2-<i>c</i>]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A

Hannes Falke, A. Chaikuad, Anja Becker et al. · Journal of Medicinal Chemistry · 2015 · 99 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Identification of 2-Anilino-9-methoxy-5,7-dihydro-6<i>H</i>-pyrimido[5,4-<i>d</i>][1]benzazepin-6-ones as Dual PLK1/VEGF-R2 Kinase Inhibitor Chemotypes by Structure-Based Lead Generation

Anne‐Marie Egert‐Schmidt, Jan Dreher, Ute Dunkel et al. · Journal of Medicinal Chemistry · 2010 · 67 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

3,6-Diamino-4-(2-halophenyl)-2-benzoylthieno[2,3-<i>b</i>]pyridine-5-carbonitriles Are Selective Inhibitors of Plasmodium falciparum Glycogen Synthase Kinase-3

Wiebke Fugel, A.E. Oberholzer, Bernhard Gschloessl et al. · Journal of Medicinal Chemistry · 2012 · 62 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +15

2-Anilino-4-(benzimidazol-2-yl)pyrimidines – A multikinase inhibitor scaffold with antiproliferative activity toward cancer cell lines

Renate Determann, Jan Dreher, Knut Baumann et al. · European Journal of Medicinal Chemistry · 2012 · 50 citations · Full text

Medicine, Medicinal Chemistry, Oncology +13

Inhibitors of the RET tyrosine kinase based on a 2-(alkylsulfanyl)-4-(3-thienyl)nicotinonitrile scaffold

Wiebke Brandt, Luca Mologni, Lutz Preu et al. · European Journal of Medicinal Chemistry · 2010 · 50 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +9