Michelle Gazdik

Inhibition of Plasmepsin V Activity Demonstrates Its Essential Role in Protein Export, PfEMP1 Display, and Survival of Malaria Parasites

Brad E. Sleebs, Sash Lopaticki, Danushka S. Marapana et al. · PLoS Biology · 2014 · 162 citations · Full text

Antiparasitic Agent, Malaria, Immunology +18

Structural basis for plasmepsin V inhibition that blocks export of malaria proteins to human erythrocytes

Anthony N. Hodder, Brad E. Sleebs, Peter E. Czabotar et al. · Nature Structural & Molecular Biology · 2015 · 109 citations

Protein Function, Biochemistry, Antiparasitic Agent +9

Pyridyl Benzamides as a Novel Class of Potent Inhibitors for the Kinetoplastid<i>Trypanosoma brucei</i>

Lori Ferrins, Michelle Gazdik, Raphaël Rahmani et al. · Journal of Medicinal Chemistry · 2014 · 58 citations

Transition State Mimetics of the <i>Plasmodium</i> Export Element Are Potent Inhibitors of Plasmepsin V from <i>P. falciparum</i> and <i>P. vivax</i>

Brad E. Sleebs, Michelle Gazdik, Matthew T. O’Neill et al. · Journal of Medicinal Chemistry · 2014 · 56 citations · Full text

Protein Function, Plasmodium Falciparum, Biochemistry +15

Novel Human Aminopeptidase N Inhibitors: Discovery and Optimization of Subsite Binding Interactions

Ji Sook Lee, Natalie B. Vinh, Nyssa Drinkwater et al. · Journal of Medicinal Chemistry · 2019 · 22 citations · Full text