Kamal Fettis

Small-molecule factor D inhibitors targeting the alternative complement pathway

Jürgen Maibaum, Sha-Mei Liao, Anna Vulpetti et al. · Nature Chemical Biology · 2016 · 74 citations · Full text

Complement System, Autoimmune Disease, Allergy +9

Trithiocarbonates as a Novel Class of HDAC Inhibitors: SAR Studies, Isoenzyme Selectivity, and Pharmacological Profiles

Florian Dehmel, Steffen Weinbrenner, Heiko Julius et al. · Journal of Medicinal Chemistry · 2008 · 40 citations · Full text

Histone Deacetylases, Hdac Inhibitors, Pharmacotherapy +17

Discovery of Highly Potent and Selective Small-Molecule Reversible Factor D Inhibitors Demonstrating Alternative Complement Pathway Inhibition <i>in Vivo</i>

Edwige Lorthiois, Karen Anderson, Anna Vulpetti et al. · Journal of Medicinal Chemistry · 2017 · 35 citations · Full text

Inflammation, Complement System, Autoimmune Disease +14

Synthesis of 3₁₀-Helix-Inducing Constrained Analogues of <scp>l</scp>-Proline

Stephen Hanessian, Gianluca Papeo, Kamal Fettis et al. · The Journal of Organic Chemistry · 2004 · 32 citations

Synthesis of Functionally Diverse and Conformationally Constrained Polycyclic Analogues of Proline and Prolinol

Stephen Hanessian, Gianluca Papeo, Mauro Angiolini et al. · The Journal of Organic Chemistry · 2003 · 24 citations

Derivatives, Heterocyclic, Biochemistry +14